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Toplam kayıt 6, listelenen: 1-6
Design and Bioevaluation of Novel Hydrazide-Hydrazones Derived from 4-Acetyl-N-Substituted Benzenesulfonamide
(Maik Nauka/Interperiodica/Springer, 2020)
In this research, a series of hydrazine-hydrazone derivatives (Ia-g), (IIa-h) were synthesized to discover new antioxidant and anticholinesterase agents. The structures of synthesized compounds were characterized by ...
Design and Antiproliferative and Antioxidant Activities of Furan-Based Thiosemicarbazides and 1,2,4-Triazoles: Their Structure-Activity Relationship and SwissADME Predictions
(Springer, 2021)
Due to the limited number of drugs in current clinical use, the diverse biological applications of furan
have encouraged the preparation of a wide variety of thiosemicarbazide and triazole derivatives for the purpose of ...
CHEMICAL COMPOSITION AND ANTIMICROBIAL ACTIVITY OF ESSENTIAL OIL OF CITRUS SINENSIS: INTERACTION WITH AMPICILLIN AND FLUCONAZOLE
(EDITURA ACAD ROMANE, 2020)
In the present study, the interactions of essential oil (EO) of Citrus sinensis L. Osbeck with two antibiotics (ampicillin and fluconazole), which are commonly used in the treatment of infections, were investigated. C. ...
Synthesis of benzoyl hydrazones having 4-hydroxy-3,5-dimethoxy phenyl ring, their biological activities, and molecular modeling studies on enzyme inhibition activities
(SCIENTIFIC TECHNICAL RESEARCH COUNCIL TURKEY-TUBITAK, 2021)
Hydrazone compounds such as anticholinesterase, tyrosinase, and urease have high capacity in terms of antioxidant activity and enzyme inhibition activities. In this study, benzoyl hydrazones compounds (7a-7m) were synthesized ...
Synthesis, predictions of drug-likeness, and pharmacokinetic properties of some chiral thioureas as potent enzyme inhibition agents
(SCIENTIFIC TECHNICAL RESEARCH COUNCIL TURKEY-TUBITAK, 2022)
A series of chiral thioureas (1 - 17) were synthesized from and tested for their anticholinesterase, tyrosinase, and urease enzyme inhibitor activities. Various phenylisothiocyanates were added to solution of ??-cysteine ...
Effects of Hypericum perforatum extract on 6-hydroxydopamine neurotoxicity in differentiated SH-SY5Y cells
(EGYPTIAN PHARMACEUTICAL JOURNAL, 2023)
Background and objectiveParkinson's disease (PD) is the second most common neurodegenerative disease after Alzheimer's disease. In our study, PD model was created as a result of exposure to 6-hydroxydopamine (6-OHDA) in ...